8PKX | pdb_00008pkx

Kelch domain of KEAP1 in complex with a ortho-dimethylbenzene linked cyclic peptide 11 (ortho-WRCNPETaEC).

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RCSB PDB Mol* Viewer 2.11.4 [4/4/2025, 6:48:47 PM]
Sequence of
     ​G​​H​​M​​K​​P​​T​​Q​​V​​M​​P​     ​S​​R​​A​​P​​K​​V​​G​​R​​L​​I​329  ​Y​​T​​A​​G​​G​​Y​​F​​R​​Q​​S​339  ​L​​S​​Y​​L​​E​​A​​Y​​N​​P​​S​349  ​D​​G​​T​​W​​L​​R​​L​​A​​D​​L​359  ​Q​​V​​P​​R​​S​​G​​L​​A​​G​​C​369  ​V​​V​​G​​G​​L​​L​​Y​​A​​V​​G​379  ​G​​R​​N​​N​​S​​P​​D​​G​​N​​T​389  ​D​​S​​S​​A​​L​​D​​C​​Y​​N​​P​399  ​M​​T​​N​​Q​​W​​S​​P​​C​​A​​P​409  ​M​​S​​V​​P​​R​​N​​R​​I​​G​​V​419  ​G​​V​​I​​D​​G​​H​​I​​Y​​A​​V​429  ​G​​G​​S​​H​​G​​C​​I​​H​​H​​N​439  ​S​​V​​E​​R​​Y​​E​​P​​E​​R​​D​449  ​E​​W​​H​​L​​V​​A​​P​​M​​L​​T​459  ​R​​R​​I​​G​​V​​G​​V​​A​​V​​L​469  ​N​​R​​L​​L​​Y​​A​​V​​G​​G​​F​479  ​D​​G​​T​​N​​R​​L​​N​​S​​A​​E​489  ​C​​Y​​Y​​P​​E​​R​​N​​E​​W​​R​499  ​M​​I​​T​​A​​M​​N​​T​​I​​R​​S​509  ​G​​A​​G​​V​​C​​V​​L​​H​​N​​C​519  ​I​​Y​​A​​A​​G​​G​​Y​​D​​G​​Q​529  ​D​​Q​​L​​N​​S​​V​​E​​R​​Y​​D​539  ​V​​A​​T​​A​​T​​W​​T​​F​​V​​A​549  ​P​​M​​K​​H​​R​​R​​S​​A​​L​​G​559  ​I​​T​​V​​H​​Q​​G​​R​​I​​Y​​V​569  ​L​​G​​G​​Y​​D​​G​​H​​T​​F​​L​579  ​D​​S​​V​​E​​C​​Y​​D​​P​​D​​T​589  ​D​​T​​W​​S​​E​​V​​T​​R​​M​​T​599  ​S​​G​​R​​S​​G​​V​​G​​V​​A​​V​609  ​T​​M​​E​​P​​S​​R​​K​​Q​​I​​D​     ​Q​​Q​​N​​S​​T​​S​
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